X0304 4 2011-09-08 0 0000880643 GENTA INC DE/ GNTA 0001100843 WARRELL RAYMOND P JR C/O GENTA INCORPORATED 200 CONNELL DRIVE BERKELEY HEIGHTS NJ 07922 1 1 0 0 Chairman & Chief Exec Officer Common Stock 2011-09-08 4 C 0 16778523 .0015 A 3462997557 D Common Stock 2011-09-21 4 S 0 8000000 0.0019 D 3454997557 D Common Stock 2011-09-22 4 S 0 8778523 0.0015 D 3446219034 D Common Stock 25170499 I By spouse 15% Senior Convertible Promissory Note 0.0015 2011-09-08 4 C 0 25000 0 A 2008-10-07 2013-09-04 Common Stock 16778523 1758468 D Includes 16,778,523 shares of common stock held jointly with Dr. Warrell's spouse, Dr. Itri, 9,237,920 shares potentially issuable upon the vesting of outstanding restricted stock units held by Dr. Warrell, 1,180,180,147 shares of common stock issuable upon the conversion of Senior Convertible Promissory Notes due Sept. 4, 2013, held in joint account, 7,010,765 shares of common stock issuable upon the conversion of Notes held by Dr. Warrell's IRA, 924,362,094 shares of common stock issuable upon the exercise of March 2010 Warrants held in joint account, 120,807,405 shares of common stock issuable upon the exercise of December 2010 Warrants held in joint account, 1,196,958,664 shares of common stock issuable upon the exercise of September 2011 Warrants held in joint account, 651,274 shares of common stock issuable upon the exercise of December 2010 Warrants held by Dr. Warrell's IRA and 7,010,765 issuable upon the exercise of September 2011 Warrants held by Dr. Warrell's IRA. Includes 3,161,191 shares of common stock potentially issuable upon the vesting of currently outstanding restricted stock units held by Dr. Itri, 10,516,174 shares of common stock issuable upon the conversion of Senior Convertible Promissory Notes due September 4, 2013, held by Dr. Itri's IRA, 976,960 shares of common stock issuable upon the exercise of December 2010 Warrants held by Dr. Itri's IRA and 10,516,174 shares of common stock issuable upon the exercise of September 2011 Warrants. Raymond P. Warrell Jr. M.D. 2011-09-23