X0303 4 2011-02-17 0 0000880643 GENTA INC DE/ GNTA 0001100843 WARRELL RAYMOND P JR C/O GENTA INCORPORATED 200 CONNELL DRIVE BERKELEY HEIGHTS NJ 07922 1 1 0 0 Chairman & Chief Exec Officer Common Stock 2011-02-17 4 S 0 820000 .0067 D 1082803801 D Common Stock 2011-02-18 4 S 0 15600 .2523 D 21640472 D Common Stock 2011-02-22 4 X 0 580000 .16 A 21094588 D Common Stock 2011-02-22 4 S 0 150000 .2532 D 20944588 D Common Stock 152695 I By spouse March 2010 Warrant 0.16 2011-02-22 4 X 0 1125884 0 D 2010-03-09 2013-03-09 Common Stock 580000 9738707 D Includes 780,000 shares of common stock held in joint account with Dr. Warrell's spouse, Dr. Itri, 5,981,681 shares of common stock potentially issuable upon the vesting of currently outstanding restricted stock units, 529,519,984 shares of common stock issuable upon the conversion of Senior Convertible Promissory Notes due September 4, 2011, as amended (the Notes), 3,032,500 shares of common stock issuable upon the conversion of Notes held by Dr. Warrell's IRA, 486,935,389 shares of common stock issuable upon the exercise of March 2010 Warrants, 56,250,980 shares of common stock issuable upon the exercise of December 2010 Warrants and 303,267 shares of common stock issuable upon the exercise of December 2010 Warrants held by Dr. Warrell's IRA. Adjusted for a 1:50 reverse stock split implemented February 18, 2011. Includes 119,632 shares of common stock potentially issuable upon the vesting of currently outstanding restricted stock units,10,590,399 shares of common stock issuable upon the conversion of Notes, 60,650 shares of common stock issuable upon the conversion of Notes held by Dr. Warrell's IRA, 9,738,707 shares of common stock issuable upon the exercise of March 2010 Warrants, 1,125,019 shares of common stock issuable upon the exercise of December 2010 Warrants and 6,065 shares of common stock issuable upon the exercise of December 2010 Warrants held by Dr. Warrell's IRA. Includes 52,622 shares of common stock potentially issuable upon the vesting of currently outstanding restricted stock units held by Dr. Itri, 90,975 shares of common stock issuable upon the conversion of Notes held by Dr. Itri and 9,098 shares of common stock issuable upon the exercise of December 2010 Warrants. These transactions were conducted under a 10b5-1 Plan, as defined under the Securities Exchange Act of 1934, as amended. /s/ Raymond P. Warrell, Jr. 2011-02-22