X0303 4 2011-01-24 0 0000880643 GENTA INC DE/ GNTA 0001100843 WARRELL RAYMOND P JR C/O GENTA INCORPORATED 200 CONNELL DRIVE BERKELEY HEIGHTS NJ 07922 1 1 0 0 Chairman & Chief Exec Officer Common Stock 2011-01-24 4 C 0 2215946 .0032 A 1095953693 D Common Stock 2011-01-25 4 S 0 2215946 .0101 D 1093737747 D Common Stock 7634855 I By spouse 15% Senior Convertible Promissory Note .0032 2011-01-24 4 C 0 7091.03 0 D 2008-10-07 2011-09-04 Common Stock 2215946 533951878 D Includes 2,215,946 shares of common stock held in joint account with Dr. Warrell's spouse, Dr. Itri, 5,981,681 shares of common stock potentially issuable upon the vesting of currently outstanding restricted stock units, 533,951,878 shares of common stock issuable upon the conversion of Senior Convertible Promissory Notes due September 4, 2011, as amended (the Notes), 3,032,500 shares of common stock issuable upon the conversion of Notes held by Dr. Warrell's IRA, 494,217,441 shares of common stock issuable upon the exercise of March 2010 Warrants, 56,250,980 shares of common stock issuable upon the exercise of December 2010 Warrants and 303,267 shares of common stock issuable upon the exercise of December 2010 Warrants held by Dr. Warrell's IRA. Includes 2,631,203 shares of common stock potentially issuable upon the vesting of currently outstanding restricted stock units held by Dr. Itri, 4,548,750 shares of common stock issuable upon the conversion of Notes held by Dr. Itri and 454,902 shares of common stock issuable upon the exercise of December 2010 Warrants. This transaction was conducted under a 10b5-1 Plan, as defined under the Securities Exchange Act of 1934, as amended. /s/ Raymond P. Warrell, Jr. 2011-01-25