X0306 4 2013-11-04 0001195116 Arno Therapeutics, Inc ARNI 0001296549 Belldegrun Arie C/O ARNO THERAPEUTICS, INC. 200 ROUTE 31 NORTH, SUITE 104 FLEMINGTON NJ 08822 1 0 0 0 Common Stock 3115 D Common Stock 143809 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust Common Stock 254887 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust Common Stock 379294 I Belldegrun Family Trust Common Stock 174644 I MDRB Partnership, L.P. Common Stock 100481 I Arie S. Belldegrun, M.D. Inc. Profit Sharing Plan Stock Option (right to buy) 19.36 2018-03-31 Common Stock 24922 24922 D Stock Option (right to buy) 8.00 2019-09-29 Common Stock 1250 1250 D Stock Option (right to buy) 8.00 2020-09-09 Common Stock 37500 37500 D Stock Option (right to buy) 8.00 2020-11-05 Common Stock 1250 1250 D Stock Option (right to buy) 2.40 2013-11-04 4 A 0 3559296 0 A 2023-11-04 Common Stock 3559296 3559296 D 2010 Class B Warrants (right to buy) 3.08 2010-09-09 2015-09-09 Common Stock 105000 105000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust 2013 Series D Warrants (right to buy) 4.00 2013-10-29 2018-10-29 Common Stock 104166 104166 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust 2013 Series E Warrants (right to buy) 2.40 2013-10-29 2014-10-31 Common Stock 104166 104166 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust 2012 Series A Warrants (right to buy) 2.40 2012-11-26 2017-11-26 Common Stock 208333 208333 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust 2012 Series B Warrants (right to buy) 2.40 2013-10-29 2014-10-31 Common Stock 125000 125000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust 2013 Series D Warrants (right to buy) 4.00 2013-10-29 2018-10-29 Common Stock 104166 104166 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust 2013 Series E Warrants (right to buy) 2.40 2013-10-29 2014-10-31 Common Stock 104166 104166 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust 2010 Class B Warrants (right to buy) 3.08 2010-09-09 2015-09-09 Common Stock 6562 6562 I Belldegrun Family Trust 2012 Series A Warrants (right to buy) 2.40 2012-11-26 2017-11-26 Common Stock 243055 243055 I Belldegrun Family Trust 2012 Series B Warrants (right to buy) 2.40 2013-10-29 2014-10-31 Common Stock 145833 145833 I Belldegrun Family Trust 2013 Series D Warrants (right to buy) 4.00 2013-10-29 2018-10-29 Common Stock 187500 187500 I Belldegrun Family Trust 2013 Series E Warrants (right to buy) 2.40 2013-10-29 2014-10-31 Common Stock 187500 187500 I Belldegrun Family Trust 2010 Class B Warrants (right to buy) 3.08 2010-09-09 2015-09-09 Common Stock 52500 52500 I MDRB Partnership, L.P. 2012 Series A Warrants (right to buy) 2.40 2012-11-26 2017-11-26 Common Stock 104166 104166 I MDRB Partnership, L.P. 2012 Series B Warrants (right to buy) 2.40 2013-10-29 2014-10-31 Common Stock 62500 62500 I MDRB Partnership, L.P. 2013 Series D Warrants (right to buy) 4.00 2013-10-29 2018-10-29 Common Stock 83333 83333 I MDRB Partnership, L.P. 2013 Series E Warrants (right to buy) 2.40 2013-10-29 2014-10-31 Common Stock 83333 83333 I MDRB Partnership, L.P. 2012 Series A Warrants (right to buy) 2.40 2012-11-26 2017-11-26 Common Stock 138888 138888 I Arie S. Belldegrun, M.D. Inc. Profit Sharing Plan 2012 Series B Warrants (right to buy) 2.40 2013-10-29 2014-10-31 Common Stock 83333 83333 I Arie S. Belldegrun, M.D. Inc. Profit Sharing Plan Although the Reporting Person is not a trustee of the BTL Trust, the Reporting Person is a beneficiary of the BTL Trust, and as such may be deemed to be the beneficial owner of the securities owned by the BTL Trust. The Reporting Person disclaims beneficial ownership of such securities except to the extent of his pecuniary interest therein. Although the Reporting Person is not a trustee of the Tampere Trust, the Reporting Person is a beneficiary of the Tampere Trust, and as such may be deemed to be the beneficial owner of the securities owned by the Tampere Trust. The Reporting Person disclaims beneficial ownership of such securities except to the extent of his pecuniary interest therein. The Reporting Person is the trustee of the family trust that owns the securities. The Reporting Person disclaims beneficial ownership of such securities except to the extent of his pecuniary interest therein. The Reporting Person is the managing partner of the limited partnership that owns the securities. The Reporting Person disclaims beneficial ownership of such securities except to the extent of his pecuniary interest therein. The Reporting Person is the trustee of the profit sharing plan that owns the securities. Currently exercisable. Vests in three equal annual installments commencing 11/5/11. Vests in equal 36-monthly installments commencing 12/4/13. /s/ Christopher J. Melsha as Attorney-in-Fact for Arie S. Belldegrun pursuant to a Power of Attorney previously filed. 2013-11-06