X0206 3 2013-01-25 0 0001195116 Arno Therapeutics, Inc ARNI 0001296549 Belldegrun Arie C/O ARNO THERAPEUTICS, INC. 200 ROUTE 31 NORTH, SUITE 104 FLEMINGTON NJ 08822 1 0 0 0 Common Stock 24922 D Common Stock 317155 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust Common Stock 127619 I Belldegrun Family Trust Common Stock 127619 I MDRB Partnership, L.P. Stock Option (right to buy) 2.42 2018-03-31 Common Stock 199377 D Stock Option (right to buy) 1.00 2019-09-29 Common Stock 10000 D Stock Option (right to buy) 1.00 2020-09-09 Common Stock 300000 D Stock Option (right to buy) 1.00 2020-11-05 Common Stock 10000 D Class A Warrants (right to buy) .5268 2010-09-09 2013-03-09 Common Stock 20000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust Class B Warrants (right to buy) .5649 2010-09-09 2015-09-09 Common Stock 105000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust 8% Senior Convertible Debentures .30 2012-11-26 2015-11-26 Common Stock 1000000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust Series A Warrants (right to buy) .50 2012-11-26 2017-11-26 Common Stock 1000000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust Series B Warrants .30 2012-11-26 2014-05-26 Common Stock 1000000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust Class A Warrants (right to buy) .5268 2010-09-09 2013-03-09 Common Stock 10000 I Belldegrun Family Trust Class B Warrants (right to buy) .5649 2010-09-09 2015-09-09 Common Stock 52500 I Belldegrun Family Trust 8% Senior Convertible Debentures .30 2012-11-26 2015-11-26 Common Stock 1166667 I Belldegrun Family Trust Series A Warrants (right to buy) .50 2012-11-26 2017-11-26 Common Stock 1166667 I Belldegrun Family Trust Series B Warrants (right to buy) .30 2012-11-26 2014-05-26 Common Stock 1166667 I Belldegrun Family Trust Class A Warrants (right to buy) .5268 2010-09-09 2013-03-09 Common Stock 10000 I MDRB Partnership, L.P. Class B Warrants (right to buy) .5649 2010-09-09 2015-09-09 Common Stock 52500 I MDRB Partnership, L.P. 8% Senior Convertible Debentures .30 2012-11-26 2015-11-26 Common Stock 500000 I MDRB Partnership, L.P. Series A Warrants (right to buy) .50 2012-11-26 2017-11-26 Common Stock 500000 I MDRB Partnership, L.P. Series B Warrants (right to buy) .30 2012-11-26 2014-05-26 Common Stock 500000 I MDRB Partnership, L.P. 8% Senior Convertible Debentures .30 2012-11-26 2015-11-26 Common Stock 666667 I Arie S. Belldegrun, M.D. Inc. Profit Sharing Plan Series A Warrants (right to buy) .50 2012-11-26 2017-11-26 Common Stock 666667 I Arie S. Belldegrun, M.D. Inc. Profit Sharing Plan Series B Warrants (right to buy) .30 2012-11-26 2014-05-26 Common Stock 666667 I Arie S. Belldegrun, M.D. Inc. Profit Sharing Plan Currently exercisable. Vests in three equal annual installments commencing 11/5/11. Although the Reporting Person is not a trustee of the BTL Trust, the Reporting Person is a beneficiary of the BTL Trust, and as such may be deemed to be the beneficial owner of the securities owned by the BTL Trust. The Reporting Person disclaims beneficial ownership of such securities except to the extent of his pecuniary interest therein. The Reporting Person is the trustee of the family trust that owns the securities. The Reporting Person disclaims beneficial ownership of such securities except to the extent of his pecuniary interest therein. The Reporting Person is the managing partner of the limited partnership that owns the securities. The Reporting Person disclaims beneficial ownership of such securities except to the extent of his pecuniary interest therein. Although the Reporting Person is not a trustee of the Tampere Trust, the Reporting Person is a beneficiary of the Tampere Trust, and as such may be deemed to be the beneficial owner of the securities owned by the Tampere Trust. The Reporting Person disclaims beneficial ownership of such securities except to the extent of his pecuniary interest therein. The Reporting Person is the trustee of the profit sharing plan that owns the securities. /s/ Arie S. Belldegrun, M.D. 2013-01-25