X0303 4 2009-09-24 0001133869 Nile Therapeutics, Inc. NLTX 0001296549 Belldegrun Arie C/O NILE THERAPEUTICS, INC. 4 WEST 4TH AVENUE, SUITE 400 SAN MATEO CA 94402 1 0 0 0 Common Stock 76935 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust Common Stock 64800 I Belldegrun Family Trust Common Stock 243200 I Arie S. Belldegrun M.D. Inc. Profit Sharing Plan Common Stock 292000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust Stock Option (Right to Buy) 1.46 2009-09-24 4 A 0 130000 0 A 2019-09-24 Common Stock 130000 130000 D Warrant (Right to Buy) 2.71 2007-09-11 2012-09-11 Common Stock 4210 4210 I Leumi Overseas Trust Corp. Ltd. as TTEE of the BTL Trust Warrant (Right to Buy) 1.25 2009-07-07 2014-07-07 Common Stock 16200 16200 I Belldegrun Family Trust Warrant (Right to Buy) 1.71 2009-07-07 2014-07-07 Common Stock 16200 16200 I Belldegrun Family Trust Warrant (Right to Buy) 2.28 2009-07-07 2014-07-07 Common Stock 32400 32400 I Belldegrun Family Trust Warrant (Right to Buy) 1.25 2009-07-07 2014-07-07 Common Stock 60800 60800 I Arie S. Belldegrun M.D. Inc. Profit Sharing Plan Warrant (Right to Buy) 1.71 2009-07-07 2014-07-07 Common Stock 60800 60800 I Arie S. Belldegrun M.D. Inc. Profit Sharing Plan Warrant (Right to Buy) 2.28 2009-07-07 2014-07-07 Common Stock 121600 121600 I Arie S. Belldegrun M.D. Inc. Profit Sharing Plan Warrant (Right to Buy) 1.25 2009-07-07 2014-07-07 Common Stock 73000 73000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust Warrant (Right to Buy) 1.71 2009-07-07 2014-07-07 Common Stock 73000 73000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust Warrant (Right to Buy) 2.28 2009-07-07 2014-07-07 Common Stock 146000 146000 I Leumi Overseas Trust Corp. Ltd. as TTEE of the Tampere Trust Although the Reporting Person is not a trustee of the BTL Trust, the Reporting Person is a beneficiary of the BTL Trust, and as such may be deemed to be the beneficial owner of the shares and the warrants owned by the BTL Trust. The Reporting Person disclaims beneficial ownership of the shares and warrants except to the extent of his pecuniary interest therein. The Reporting Person is the Trustee of the family trust that owns the shares and the warrants. The Reporting Person disclaims beneficial ownership of these shares and warrants except to the extent of his pecuniary interest therein. The Reporting Person is the Trustee of the profit sharing plan that owns the shares and the warrants. Although the Reporting Person is not a trustee of the Tampere Trust, the Reporting Person is a beneficiary of the Tampere Trust, and as such may be deemed to be the beneficial owner of the shares and the warrants owned by the Tampere Trust. The Reporting Person disclaims beneficial ownership of the shares and warrants except to the extent of his pecuniary interest therein. The shares subject to the option vest in three equal installments on September 24, 2011, September 24, 2012, and September 24, 2013. /s/ Daron Evans as Attorney-in-Fact pursuant to Power of Attorney previously filed. 2009-09-28